List of cardiac pharmaceutical agents
Cardiac Pharmaceutical Agents: A Comprehensive Overview
Cardiac pharmaceutical agents are a diverse group of medications formulated to manage and treat cardiovascular diseases. These agents play a crucial role in regulating heart rate, treating arrhythmias, managing blood pressure, and other essential cardiac functions.
Classification of Cardiac Agents
Cardiac pharmaceutical agents can be categorized based on their mechanism of action and primary indications.
Antiarrhythmic Agents
Antiarrhythmic agents are designed to correct abnormal heart rhythms.
Type I: Sodium Channel Blockers
- Type Ia:
- Type Ib:
- Type Ic:
Type II: Beta Blockers
Type III: Potassium Channel Blockers
Type IV: Slow Calcium Channel Blockers
Type V: Miscellaneous
ACE Inhibitors
Angiotensin-converting enzyme (ACE) inhibitors are primarily used for treating high blood pressure and heart failure.
Angiotensin II Receptor Antagonists
These drugs block the effects of angiotensin, reducing blood pressure.
Beta Blockers
- Note: Metoprolol, previously mentioned, is also classified under this category.
Calcium Channel Blockers
- Note: Diltiazem and Verapamil, mentioned earlier, also fall into this category.
Alphabetic list of cardiac drugs
- 2-Methoxyestradiol
- 2-Methoxyestriol
- 4-Aminopyridine
- 4-Methylpregabalin
- ACE inhibitor
- ACE inhibitor and thiazide combination
- AH-1058
- AZD1305
- Abanoquil
- Abediterol
- Abitesartan
- Abnormal cannabidiol
- Acebutolol
- Acecainide
- Acefylline clofibrol
- Acepromazine
- Acetazolamide
- Acetergamine
- Acetildenafil
- Acetiromate
- Acetohexamide
- Acetryptine
- Acetyldigitoxin
- Acipimox
- Actisomide
- Adaprolol
- Adderall
- Adenosine
- Adibendan
- Adimolol
- Adrenaline
- Adrenergic antagonist
- Afurolol
- Aildenafil
- Ajmalicine
- Ajmaline
- Alacepril
- Alcohol (drug)
- Alfuzosin
- Alinidine
- Alirocumab
- Aliskiren
- Aliskiren/amlodipine
- Aliskiren/amlodipine/hydrochlorothiazide
- Aliskiren/hydrochlorothiazide
- Almokalant
- Alpha blocker
- Alpha-1 blocker
- Alpha-2 blocker
- Alpha-Methylhistamine
- Alprenolol
- Alprenoxime
- Altizide
- Aluminium clofibrate
- Aluminium nicotinate
- Amesergide
- Amezinium metilsulfate
- Amidephrine
- Amifampridine
- Amiloride
- Aminometradine
- Amiodarone
- Amitriptyline
- Amlodipine
- Amlodipine/atorvastatin
- Amlodipine/benazepril
- Amlodipine/celecoxib
- Amlodipine/valsartan
- Amosulalol
- Amoxapine
- Amphetamine
- Amrinone
- Amyl nitrite
- Ancarolol
- Angiotensin II (medication)
- Angiotensin II receptor blocker
- Angiotensinamide
- Anipamil
- Anisodamine
- Anisodine
- Anti-cholesterol
- Antianginal
- Antiarin
- Antiarrhythmic agent
- Antihistamine
- Antihypertensive drug
- Antihypotensive agent
- Antimineralocorticoid
- Apararenone
- ApoA-1 Milano
- Apomorphine
- Aprindine
- Aptazapine
- Aquaretic
- Aranidipine
- Arbaclofen placarbil
- Arbutamine
- Arenobufagin
- Arformoterol
- Aripiprazole
- Arnolol
- Arotinolol
- Arteriolar vasodilator
- Asenapine
- Asocainol
- Astemizole
- Asthmador
- Atagabalin
- Atenolol
- Atenolol/chlorthalidone
- Atipamezole
- Atiprosin
- Atomoxetine
- Atorvastatin
- Avanafil
- Azacosterol
- Azalanstat
- Azapetine
- Azaspiracid
- Azelnidipine
- Azepindole
- Azilsartan
- Azimilide
- Azosemide
- BQ-788
- BRL-32872
- BRL-44408
- Baclofen
- Bambuterol
- Bamethan
- Bamifylline
- Barbiturate
- Barnidipine
- Bay K8644
- Befunolol
- Bempedoic acid
- Bempedoic acid/ezetimibe
- Benazepril
- Bencyclane
- Bendroflumethiazide
- Benfluorex
- Benidipine
- Benoxathian
- Benzamidenafil
- Benzamil
- Benziodarone
- Benzocaine
- Benzoctamine
- Benzthiazide
- Benzylpiperazine
- Bepridil
- Berbamine
- Beta blocker
- Beta-2 adrenergic antagonist
- Beta-3 adrenergic antagonist
- Beta1-adrenergic agonist
- Beta2-adrenergic agonist
- Betahistine
- Betaxolol
- Bethanidine
- Bevantolol
- Bezafibrate
- BgK
- Bietaserpine
- Bile acid sequestrant
- Bimakalim
- Bimatoprost/timolol
- Bisoprolol
- Bitolterol
- BmP02
- Bococizumab
- Bopindolol
- Bornaprolol
- Brefonalol
- Bretylium
- Brexpiprazole
- Brinzolamide
- Brinzolamide/brimonidine
- Bromoacetylalprenololmenthane
- Broxaterol
- Bucindolol
- Bucladesine
- Bucumolol
- Budiodarone
- Budralazine
- Bufadienolide
- Bufagin
- Bufalin
- Bufanolide
- Bufetolol
- Buflomedil
- Bufotalin
- Bufuralol
- Bumetanide
- Bunaftine
- Bunazosin
- Bunitrolol
- Buphenine
- Bupicomide
- Bupranolol
- Buprenorphine
- Bupropion/zonisamide
- Buspirone
- Buspirone/testosterone
- Butalamine
- Butantoxin
- Butaxamine
- Butidrine
- Butizide
- Butofilolol
- Butriptyline
- Butyl nitrite
- Butynamine
- CETP inhibitor
- CGMP-specific phosphodiesterase type 5
- CGS-15943
- CXL 1020
- CYT006-AngQb
- Cadralazine
- Cafaminol
- Cafedrine
- Caffeine
- Calcium
- Calcium channel blocker
- Calcium channel blocker toxicity
- Calliotoxin
- Calotropin
- Cambiogenplasmid
- Canadine
- Candesartan
- Canrenone
- Capsinolol
- Captopril
- Caramiphen
- Carazolol
- Carbocromen
- Carbonic anhydrase inhibitor
- Carboxyamidotriazole
- Carbutamide
- Carbuterol
- Cardenolide
- Cardiac Arrhythmia Suppression Trial
- Cardiac glycoside
- Cardiac stimulant
- Cariporide
- Carmoterol
- Carpindolol
- Carpronium chloride
- Carteolol
- Carvedilol
- Casuarinin
- Cathinone
- Celiprolol
- Celivarone
- Cenderitide
- Cerberin
- Cerivastatin
- Ceronapril
- Cetamolol
- Cetiedil
- Charybdotoxin
- Chloracyzine
- Chlorisondamine
- Chlormerodrin
- Chloroethylclonidine
- Chlorophenylbiguanide
- Chloroquine
- Chlorothiazide
- Chlorphenamine
- Chlorpromazine
- Chlorpropamide
- Chlorprothixene
- Chlortalidone
- Cholesterol absorption inhibitor
- Chronotropic
- Cibenzoline
- Ciclafrine
- Cicletanine
- Ciclonicate
- Cicloprolol
- Cicutoxin
- Cilazapril
- Cilnidipine
- Cilostazol
- Cimlanod
- Cinaciguat
- Cinamolol
- Cinepazet
- Cinobufagin
- Ciprofibrate
- Cirazoline
- Cisapride
- Clazosentan
- Clenbuterol
- Clentiazem
- Clevidipine
- Clinofibrate
- Clofenamide
- Clofibrate
- Clofibric acid
- Clofibride
- Clofilium
- Clomestrone
- Clomipramine
- Clonidine
- Clopamide
- Cloperastine
- Cloranolol
- Clorexolone
- Cloridarol
- Clozapine
- Co-amilofruse
- Co-amilozide
- Co-tenidone
- Cocaine
- Colesevelam
- Colestilan
- Colestipol
- Colestolone
- Colestyramine
- Colextran
- Colterol
- Conivaptan
- Convallamarin
- Convallarin
- Convallatoxin
- Coronaridine
- Corynanthine
- Creatinolfosfate
- Cromakalim
- Cryptenamine
- Cyamemazine
- Cyanopindolol
- Cyclandelate
- Cycleanine
- Cyclohexyl nitrite
- Cyclopenthiazide
- Cyclothiazide
- Cymarin
- Cyproheptadine
- DMPX
- DSP-2230
- Daflon
- Daigremontianin
- Dalbraminol
- Dapiprazole
- Darapladib
- Darodipine
- Darusentan
- Dauricine
- Debrisoquine
- Decarbamoylsaxitoxin
- Delapril
- Dendrotoxin
- Denopamine
- Desacetylmetipranolol
- Deserpidine
- Desipramine
- Deslanoside
- Devapamil
- Dextroamphetamine
- Dextropropoxyphene
- Dextrothyroxine
- Diacetolol
- Diazoxide
- Dichloroisoprenaline
- Dicirenone
- Diclofenamide
- Diethylene glycol dinitrate
- Digitalis
- Digitoxigenin
- Digitoxin
- Digoxigenin
- Digoxin
- Dihydralazine
- Dihydrexidine
- Dihydroalprenolol
- Dihydroergocornine
- Dihydroergocristine
- Dihydroergotamine
- Dihydropyridine calcium channel blockers
- Dilazep
- Diltiazem
- Dimeditiapramine
- Dimetofrine
- Diprafenone
- Diproteverine
- Discovery and development of ACE inhibitors
- Discovery and development of angiotensin receptor blockers
- Discovery and development of beta-blockers
- Discovery and development of beta2 agonists
- Discovery and development of phosphodiesterase 5 inhibitors
- Discovery and development of statins
- Disopyramide
- Diuretic
- Dobutamine
- Dofetilide
- Domesticine
- Domperidone
- Dopamine
- Dopamine (medication)
- Dopexamine
- Dorzolamide
- Dosulepin
- Dotarizine
- Doxazosin
- Doxepin
- Draquinolol
- Dronedarone
- Droperidol
- E-4031
- Ecastolol
- Efaroxan
- Efloxate
- Efonidipine
- Emopamil
- Enalapril
- Enalapril/hydrochlorothiazide
- Enalaprilat
- Encainide
- Endothelin receptor antagonist
- Endothelium-derived hyperpolarizing factor
- Endralazine
- Enoximone
- Enpiperate
- Epanolol
- Epithelial sodium channel blocker
- Epitizide
- Eprosartan
- Ergine
- Ergotamine
- Ergovaline
- Ergtoxin
- Ericolol
- Ersentilide
- Esaxerenone
- Esmirtazapine
- Esmolol
- Etacrynic acid
- Etafenone
- Ethacizine
- Ethanolamine-O-sulfate
- Ethoxzolamide
- Ethyl eicosapentaenoic acid
- Ethyl nitrite
- Ethylene glycol dinitrate
- Etilefrine
- Etofibrate
- Etofylline nicotinate
- Etoperidone
- Etozolin
- Eugenodilol
- Evacetrapib
- Evenamide
- Evinacumab
- Evolocumab
- Exaprolol
- Ezetimibe
- Ezetimibe/atorvastatin
- Ezetimibe/rosuvastatin
- Ezetimibe/simvastatin
- F15845
- Falintolol
- Falipamil
- Fantofarone
- Fatty acid oxidation inhibitors
- Felodipine
- Felypressin
- Fendiline
- Fenmetozole
- Fenofibrate
- Fenofibrate/pravastatin
- Fenofibrate/simvastatin
- Fenoterol
- Fenquizone
- Fenspiride
- Fentanyl
- Fibrate
- Fimasartan
- Flecainide
- Flestolol
- Flosequinan
- Fluasterone
- Flunarizine
- Fluocinolone acetonide
- Fluocortolone
- Fluorometholone
- Fluparoxan
- Fluphenazine
- Flusoxolol
- Fluticasone furoate/umeclidinium bromide/vilanterol
- Fluticasone furoate/vilanterol
- Fluvastatin
- Forasartan
- Formoterol
- Fosinopril
- Funapide
- Furosemide
- Gabapentin
- Gabapentin enacarbil
- Gabapentinoid
- Gallopamil
- Gambierol
- Gamma-Glutamylmethylamide
- Gapicomine
- Gemfibrozil
- Gemopatrilat
- Gepirone
- Gitoformate
- Glibenclamide
- Glibornuride
- Glicaramide
- Gliclazide
- Glimepiride
- Glipizide
- Gliquidone
- Glisoxepide
- Glucagon (medication)
- Glyclopyramide
- Glycopyrronium bromide/formoterol
- Granatin B
- Grepafloxacin
- Guanabenz
- Guanadrel
- Guanazodine
- Guanfacine
- Guanoclor
- Guanoxabenz
- Guanoxan
- HBI-3000
- HDL-Atherosclerosis Treatment Study
- HMR 1883
- Heart Protection Study
- Heptaminol
- Hexobendine
- Hidrosmin
- Histamine
- Homosildenafil
- Hydracarbazine
- Hydralazine
- Hydralazine/isosorbide dinitrate
- Hydrazinophthalazine
- Hydrochlorothiazide
- Hydrochlorothiazide/triamterene
- Hydroflumethiazide
- Hydroxycarteolol
- Hydroxychloroquine
- Hydroxynefazodone
- Hydroxytertatolol
- Hydroxyzine
- Hypokalemic sensory overstimulation
- ICI-118,551
- Ibogaine
- Ibrolipim
- Ibutilide
- Icariin
- Idazoxan
- Idropranolol
- Ifenprodil
- Imagabalin
- Imepitoin
- Imidapril
- Imiloxan
- Imipramine
- Imolamine
- Inclisiran
- Indacaterol
- Indacaterol/mometasone
- Indacrinone
- Indane-5-sulfonamide
- Indapamide
- Indecainide
- Indenolol
- Indopanolol
- Indoramin
- Inositol nicotinate
- Inotrope
- Iodocyanopindolol
- Iodopindolol
- Iprocrolol
- Ipsapirone
- Irampanel
- Irbesartan
- Isamoltane
- Isobutyl nitrite
- Isoprenaline
- Isopropyl nitrite
- Isosorbide
- Isosorbide dinitrate
- Isosorbide mononitrate
- Isoxaprolol
- Isoxsuprine
- Isradipine
- Itramin tosilate
- Ivabradine
- JTV-519
- JUPITER trial
- K-Strophanthidin
- Kava
- Kavain
- Ketanserin
- Ketocaine
- L-163,491
- L-765,314
- Labetalol
- Lacidipine
- Lacosamide
- Lactotripeptides
- Lanatoside C
- Landiolol
- Lapaquistat
- Leconotide
- Lercanidipine
- Levacetylmethadol
- Levamlodipine
- Levoamphetamine
- Levobetaxolol
- Levobunolol
- Levomoprolol
- Levosalbutamol
- Levosimendan
- Lidanserin
- Lidocaine
- Lidoflazine
- Linopirdine
- Linsidomine
- Lipid-lowering agent
- Lisdexamfetamine
- Lisinopril
- Lisinopril/amlodipine
- Lisinopril/hydrochlorothiazide
- List of side effects of digoxin
- Lisuride
- Lixivaptan
- Lodenafil
- Lofepramine
- Lofexidine
- Lomerizine
- Lomitapide
- Long-acting beta-adrenoceptor agonist
- Loop diuretic
- Loperamide
- Lorajmine
- Lorazepam
- Lorcainide
- Losartan
- Losartan/hydrochlorothiazide
- Lovastatin
- Loxapine
- Lubazodone
- Lurasidone
- Mafenide
- Magnesium citrate
- Magnesium pyridoxal 5-phosphate glutamate
- Manidipine
- Mannitol
- Manoalide
- Maprotiline
- Marinobufagenin
- Mebutizide
- Medroxalol
- Mefruside
- Meglutol
- Meldonium
- Melperone
- Mephedrone
- Mephentermine
- Mepindolol
- Mepiprazole
- Meralluride
- Mercurial diuretic
- Mercury(I) chloride
- Mersalyl
- Meta-Chlorophenylpiperazine
- Meta-Hydroxynorephedrine
- Metahexamide
- Metaraminol
- Metazosin
- Methadone
- Methamphetamine
- Methazolamide
- Methoserpidine
- Methoxamine
- Methoxyphenamine
- Methyclothiazide
- Methyl nitrite
- Methyldopa
- Methylphenidate
- Methysticin
- Meticrane
- Metildigoxin
- Metipranolol
- Metirosine
- Metitepine
- Metolazone
- Metoprolol
- Mevastatin
- Mexiletine
- Mexrenone
- Mianserin
- Mibefradil
- Midodrine
- Milrinone
- Minoxidil
- Mipomersen
- Mirodenafil
- Mirogabalin
- Mirtazapine
- Mitiglinide
- Moexipril
- Molsidomine
- Monacolin J
- Monatepil
- Monoethanolamine oleate
- Monoxerutin
- Moprolol
- Moracizine
- Moxisylyte
- Moxonidine
- Mozavaptan
- Muzolimine
- Mytatrienediol
- N6-Cyclopentyladenosine
- NAN-190
- Nadolol
- Nadoxolol
- Nafenopin
- Naftidrofuryl
- Naftopidil
- Nantenine
- Naphazoline
- Nateglinide
- Nebivolol
- Nefazodone
- Nefopam
- Neldazosin
- Neoconvalloside
- Neosaxitoxin
- Nepicastat
- Nesiritide
- Niacin
- Niacin/lovastatin
- Niacin/simvastatin
- Niaprazine
- Nicardipine
- Nicergoline
- Niceritrol
- Nicofuranose
- Nicorandil
- Nicotinic antagonist
- Nicotinyl alcohol
- Nifedipine
- Nifekalant
- Nifenalol
- Niflumic acid
- Niguldipine
- Niludipine
- Nilvadipine
- Nimodipine
- Nipradilol
- Niravoline
- Nisoldipine
- Nitrendipine
- Nitroarginine
- Nitroglycerin (medication)
- Nitrosoprodenafil
- Nitrovasodilator
- Norclomipramine
- Nordoxepin
- Norepinephrine (medication)
- Norfenefrine
- Noribogaine
- Norpropoxyphene
- Norpropylhexedrine
- Northiaden
- Nortriptyline
- Norverapamil
- Ocaperidone
- Olanzapine
- Olanzapine/samidorphan
- Oleandrin
- Olmesartan
- Olmesartan/amlodipine
- Olmesartan/amlodipine/hydrochlorothiazide
- Olmesartan/hydrochlorothiazide
- Olodaterol
- Olprinone
- Omapatrilat
- Omecamtiv mecarbil
- Omega-3 acid ethyl esters
- Omega-3 carboxylic acids
- Opipramol
- Orphenadrine
- Osmotic diuretic
- Ouabain
- Oxetacaine
- Oxetorone
- Oxodipine
- Oxprenolol
- Oxyfedrine
- Oxymetazoline
- Ozolinone
- PD-217,014
- PDE3 inhibitor
- PDE5 inhibitor
- PF-05089771
- PF-610355
- Pacrinolol
- Pafenolol
- Paliperidone
- Pamabrom
- Pamatolol
- Pamicogrel
- Papaverine
- Pardoprunox
- Pargolol
- Pargyline
- Pedunculagin
- Pelanserin
- Pemafibrate
- Penbutolol
- Pentaerythritol tetranitrate
- Pentifylline
- Pentolinium
- Pentoxifylline
- Perhexiline
- Perindopril
- Perindopril/indapamide
- Perlapine
- Peruvoside
- Pethidine
- PhTx-1
- Phendioxan
- Phenibut
- Phenoxybenzamine
- Phentolamine
- Phenylephrine
- Phenylephrine/ketorolac
- Phenytoin
- Phytosterol
- Pildralazine
- Pilsicainide
- Pimobendan
- Pimozide
- Pinacidil
- Pinaverium bromide
- Pindobind
- Pindolol
- Pipamperone
- Piperoxan
- Pirbuterol
- Piretanide
- Piribedil
- Pirolazamide
- Pitavastatin
- Pizotifen
- Polidocanol
- Polycap
- Polythiazide
- Poppers
- Potassium canrenoate
- Potassium channel blocker
- Potassium-sparing diuretic
- Practolol
- Prajmaline
- Pranidipine
- Pravastatin
- Prazosin
- Prednazoline
- Pregabalin
- Prenalterol
- Prenylamine
- Primidolol
- Primidone
- Proarrhythmic agent
- Procainamide
- Procaine
- Procaterol
- Procinolol
- Profenamine
- Progesterone (medication)
- Promethazine
- Pronethalol
- Propafenone
- Propatylnitrate
- Propranolol
- Propylene glycol dinitrate
- Propylhexedrine
- Prorenone
- Proroxan
- Proscillaridin
- Protriptyline
- Punicalagin
- Punicalin
- Pyrimidinylpiperazine
- Quazinone
- Quetiapine
- Quifenadine
- Quinapril
- Quinaprilat
- Quinazosin
- Quinethazone
- Quinidine
- RPL-554
- Racemorphan
- Ractopamine
- Ralfinamide
- Ramipril
- Ranolazine
- Rauwolscine
- Reboxetine
- Regadenoson
- Remacemide
- Remikiren
- Renin inhibitor
- Rentiapril
- Repaglinide
- Rescinnamine
- Reserpine
- Rhynchophylline
- Ridazolol
- Rilmenidine
- Riociguat
- Riodipine
- Risperidone
- Ritodrine
- Rolofylline
- Ronactolol
- Ronifibrate
- Rostafuroxin
- Rosuvastatin
- Rotigaptide
- Rotigotine
- Roxibolone
- Rufinamide
- S-Ethylisothiouronium diethylphosphate
- S32212
- SB-269970
- SC-8109
- SCH 900271
- SCH-48461
- SCH-58261
- SKF-83,959
- SR 59230A
- Sacubitril
- Sacubitril/valsartan
- Sacubitrilat
- Safinamide
- Salmeterol
- Satavaptan
- Saxitoxin
- Scilliroside
- Selexipag
- Sematilide
- Serelaxin
- Sertindole
- Sesamodil
- Setiptiline
- Sildenafil
- Silodosin
- Simfibrate
- Simvastatin
- Sodium apolate
- Sodium channel blocker
- Sodium nitroprusside
- Sodium tetradecyl sulfate
- Solpecainol
- Soquinolol
- Sorbitol
- Sotalol
- Sparteine
- Spegatrine
- Spiperone
- Spirapril
- Spiraprilat
- Spirendolol
- Spiroxasone
- Spiroxatrine
- Ssm spooky toxin
- Statin
- Sulfinalol
- Sulfoaildenafil
- Sulmazole
- Suloctidil
- Sultiame
- Sunepitron
- Sympatholytic
- Syrosingopine
- TROX-1
- Tadalafil
- Talinolol
- Talipexole
- Tamsulosin
- Tandospirone
- Tasosartan
- Tazolol
- Tedisamil
- Telmisartan
- Telmisartan/hydrochlorothiazide
- Temocapril
- Terazosin
- Terbutaline
- Terfenadine
- Terguride
- Terlipressin
- Tertatolol
- Tetrahydropalmatine
- Tetrandrine
- Tetrodotoxin
- Tetryzoline
- Tezosentan
- Theodrenaline
- Theophylline
- Thevetin
- Thiazide
- Thiazide-like diuretic
- Thioridazine
- Tiadenol
- Tiamenidine
- Tibric acid
- Tienilic acid
- Tienoxolol
- Tilisolol
- Timolol
- Tiodazosin
- Tiotixene
- Tipepidine
- Tiprenolol
- Tirabrutinib
- Tiracizine
- Tocainide
- Tolamolol
- Tolazamide
- Tolazoline
- Tolbutamide
- Toliprolol
- Tolonidine
- Tolperisone
- Tolvaptan
- Topiramate
- Torasemide
- Torcetrapib
- Trandolapril
- Trandolapril/verapamil
- Trapidil
- Trazodone
- Triamterene
- Triazoledione
- Tribenoside
- Trichlormethiazide
- Trimazosin
- Trimecaine
- Trimetazidine
- Trimipramine
- Tripamide
- Triparanol
- Trolnitrate
- Troxerutin
- Tst26
- Udenafil
- Ulimorelin
- Umeclidinium bromide/vilanterol
- Urapidil
- Valsartan
- Valsartan/hydrochlorothiazide
- Vardenafil
- Vasoconstriction
- Vasoprotective
- Venalex
- Verapamil
- Vericiguat
- Vermistatin
- Vernakalant
- Verrucotoxin
- Versutoxin
- Vesnarinone
- Vilanterol
- Vinburnine
- Vinpocetine
- Visnadine
- Vixotrigine
- Voacangine
- Volanesorsen
- WB-4101
- XEN-D0101
- Xamoterol
- Xanthinol
- Xibenolol
- Xipamide
- Xipranolol
- Xylometazoline
- Yohimbine
- Zaprinast
- Zetekitoxin AB
- Ziconotide
- Zilpaterol
- Zofenopril
- Zofenoprilat
- Zolertine
- Zonisamide
- Zotepine
- Α-Acetyldigoxin
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