Carpindolol
| Carpindolol | |
|---|---|
| Carpindolol.svg | |
| INN | |
| Drug class | |
| Routes of administration | |
| Pregnancy category | |
| Bioavailability | |
| Metabolism | |
| Elimination half-life | |
| Excretion | |
| Legal status | |
| CAS Number | |
| PubChem | |
| DrugBank | |
| ChemSpider | |
| KEGG | |
Carpindolol is a beta-blocker medication used primarily in the treatment of hypertension and certain types of cardiac arrhythmias. It is known for its ability to block beta-adrenergic receptors, which are part of the sympathetic nervous system.
Pharmacology[edit]
Carpindolol functions by inhibiting the action of epinephrine and norepinephrine on beta-adrenergic receptors. This leads to a decrease in heart rate, cardiac output, and blood pressure. The drug is classified as a non-selective beta-blocker, meaning it affects both beta-1 and beta-2 receptors.
Mechanism of Action[edit]
Carpindolol binds to beta-adrenergic receptors on the surface of cells in the heart and vascular smooth muscle. By blocking these receptors, it prevents the usual binding of catecholamines, which are responsible for increasing heart rate and force of contraction. This results in a reduction of myocardial oxygen demand and a decrease in blood pressure.
Clinical Uses[edit]
Carpindolol is primarily used in the management of:
Side Effects[edit]
Common side effects of Carpindolol include:
Less common but more serious side effects can include:
Contraindications[edit]
Carpindolol should not be used in patients with:
Related pages[edit]
Medical Disclaimer: WikiMD is for informational purposes only and is not a substitute for professional medical advice. Content may be inaccurate or outdated and should not be used for diagnosis or treatment. Always consult your healthcare provider for medical decisions. Verify information with trusted sources such as CDC.gov and NIH.gov. By using this site, you agree that WikiMD is not liable for any outcomes related to its content. See full disclaimer.
Credits:Most images are courtesy of Wikimedia commons, and templates, categories Wikipedia, licensed under CC BY SA or similar.
Translate this page: - East Asian
中文,
日本,
한국어,
South Asian
हिन्दी,
தமிழ்,
తెలుగు,
Urdu,
ಕನ್ನಡ,
Southeast Asian
Indonesian,
Vietnamese,
Thai,
မြန်မာဘာသာ,
বাংলা
European
español,
Deutsch,
français,
Greek,
português do Brasil,
polski,
română,
русский,
Nederlands,
norsk,
svenska,
suomi,
Italian
Middle Eastern & African
عربى,
Turkish,
Persian,
Hebrew,
Afrikaans,
isiZulu,
Kiswahili,
Other
Bulgarian,
Hungarian,
Czech,
Swedish,
മലയാളം,
मराठी,
ਪੰਜਾਬੀ,
ગુજરાતી,
Portuguese,
Ukrainian