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Template
:
Histamine receptor modulators
From WikiMD's Wellness Encyclopedia
Revision as of 19:46, 25 July 2022 by
en>Frietjes
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Histamine receptor
modulators
H
1
Agonists
*
2-Pyridylethylamine
Betahistine
Histamine
HTMT
L
-Histidine
UR-AK49
Antagonists
*
First-generation:
4-Methyldiphenhydramine
Alimemazine
Antazoline
Azatadine
Bamipine
Benzatropine (benztropine)
Bepotastine
Bromazine
Brompheniramine
Buclizine
Captodiame
Carbinoxamine
Chlorcyclizine
Chloropyramine
Chlorothen
Chlorphenamine
Chlorphenoxamine
Cinnarizine
Clemastine
Clobenzepam
Clocinizine
Cloperastine
Cyclizine
Cyproheptadine
Dacemazine
Decloxizine
Deptropine
Dexbrompheniramine
Dexchlorpheniramine
Dimenhydrinate
Dimetindene
Diphenhydramine
Diphenylpyraline
Doxylamine
Embramine
Etodroxizine
Etybenzatropine (ethylbenztropine)
Etymemazine
Fenethazine
Flunarizine
Histapyrrodine
Homochlorcyclizine
Hydroxyethylpromethazine
Hydroxyzine
Isopromethazine
Isothipendyl
Meclozine
Medrylamine
Mepyramine (pyrilamine)
Mequitazine
Methafurylene
Methapyrilene
Methdilazine
Moxastine
Orphenadrine
Oxatomide
Oxomemazine
Perlapine
Phenindamine
Pheniramine
Phenyltoloxamine
Pimethixene
Piperoxan
Pipoxizine
Promethazine
Propiomazine
Pyrrobutamine
Talastine
Thenalidine
Thenyldiamine
Thiazinamium
Thonzylamine
Tolpropamine
Tripelennamine
Triprolidine
Second/third-generation:
Acrivastine
Alinastine
Astemizole
Azelastine
Bamirastine
Barmastine
Bepiastine
Bepotastine
Bilastine
Cabastinen
Carebastine
Cetirizine
Clemastine
Clemizole
Clobenztropine
Desloratadine
Dorastine
Ebastine
Efletirizine
Emedastine
Epinastine
Fexofenadine
Flezelastine
Ketotifen
Latrepirdine
Levocabastine
Levocetirizine
Linetastine
Loratadine
Mapinastine
Mebhydrolin
Mizolastine
Moxastine
Noberastine
Octastine
Olopatadine
Perastine
Pibaxizine
Piclopastine
Quifenadine (phencarol)
Rocastine
Rupatadine
Setastine
Sequifenadine (bicarphen)
Talastine
Temelastine
Terfenadine
Vapitadine
Zepastine
Others:
Atypical antipsychotics
(e.g.,
aripiprazole
,
asenapine
,
brexpiprazole
,
brilaroxazine
,
clozapine
,
iloperidone
,
olanzapine
,
paliperidone
,
quetiapine
,
risperidone
,
ziprasidone
,
zotepine
)
Phenylpiperazine
antidepressants
(e.g.,
hydroxynefazodone
,
nefazodone
,
trazodone
,
triazoledione
)
Tetracyclic antidepressants
(e.g.,
amoxapine
,
loxapine
,
maprotiline
,
mianserin
,
mirtazapine
,
oxaprotiline
)
Tricyclic antidepressants
(e.g.,
amitriptyline
,
butriptyline
,
clomipramine
,
desipramine
,
dosulepin (dothiepin)
,
doxepin
,
imipramine
,
iprindole
,
lofepramine
,
nortriptyline
,
protriptyline
,
trimipramine
)
Typical antipsychotics
(e.g.,
chlorpromazine
,
flupenthixol
,
fluphenazine
,
loxapine
,
perphenazine
,
prochlorperazine
,
thioridazine
,
thiothixene
)
Unknown/unsorted:
Azanator
Belarizine
Elbanizine
Flotrenizine
GSK1004723
Napactadine
Tagorizine
Trelnarizine
Trenizine
H
2
Agonists
*
Amthamine
Betazole
Dimaprit
Histamine
HTMT
Impromidine
L
-Histidine
UR-AK49
Antagonists
*
Bisfentidine
Burimamide
Cimetidine
Dalcotidine
Donetidine
Ebrotidine
Etintidine
Famotidine
Isolamtidine
Lafutidine
Lamtidine
Lavoltidine (loxtidine)
Lupitidine
Metiamide
Mifentidine
Niperotidine
Nizatidine
Osutidine
Oxmetidine
Pibutidine
Quisultazine (quisultidine)
Ramixotidine
Ranitidine
Roxatidine
Sufotidine
Tiotidine
Tuvatidine
Venritidine
Xaltidine
Zolantidine
H
3
Agonists
*
α-Methylhistamine
Cipralisant
Histamine
Imetit
Immepip
Immethridine
L
-Histidine
Methimepip
Proxyfan
Antagonists
*
A-349821
A-423579
ABT-239
ABT-652
AZD5213
Bavisant
Betahistine
Burimamide
Ciproxifan
Clobenpropit
Conessine
Enerisant
GSK-189254
Impentamine
Iodophenpropit
Irdabisant
JNJ-5207852
NNC 38-1049
PF-03654746
Pitolisant
SCH-79687
Thioperamide
VUF-5681
H
4
Agonists
*
4-Methylhistamine
α-Methylhistamine
Histamine
L
-Histidine
OUP-16
VUF-8430
Antagonists
*
JNJ-7777120
Mianserin
Seliforant
Thioperamide
Toreforant
VUF-6002
;See also
Receptor/signaling modulators
Monoamine metabolism modulators
Monoamine reuptake inhibitors
Category
:
Drug templates by receptor, channel, or pump