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Template:Pharmacomodulation

From WikiMD's Wellness Encyclopedia

Pharmacomodulation
Types
* ♦ Enzyme: Inducer
  • Inhibitor
  • ♦ Ion channel: Opener
  • Blocker
  • ♦ Receptor: Agonist
  • Partial agonist
  • Antagonist
  • Inverse agonist
  • Positive allosteric modulator (PAM)
  • Negative allosteric modulator (NAM)
  • ♦ Transporter [Reuptake vs Efflux]: Enhancer (RE)
  • Inhibitor (RI)
  • Releaser (RA)
  • ♦ Miscellaneous: Precursor
  • Cofactor
Classes
Enzyme
see Enzyme inhibition
Ion channel
See Ion channel modulators
Receptor &
transporter
BA/M
Adrenergic
* Adrenergic receptor agonist (α
  • β (1
  • 2))
  • Adrenergic receptor antagonist (α (1
  • 2)
  • β)
  • Norepinephrine reuptake inhibitor (NRI)
Dopaminergic
* Dopamine receptor agonist
  • Dopamine receptor antagonist
  • Dopamine reuptake inhibitor (DRI)
Histaminergic
* Histamine receptor agonist
  • Histamine receptor antagonist (H1
  • H2
  • H3)
AA
Cholinergic
* Acetylcholine receptor agonist (Muscarinic
  • Nicotinic)
    • Cholinesterase inhibitor
  • Acetylcholine receptor antagonist (Muscarinic
  • Nicotinic (Ganglionic
  • Muscular))
Cannabinoidergic
* Cannabinoid receptor agonist
  • Cannabinoid receptor antagonist
  • Endocannabinoid enhancer (eCBE)
  • Endocannabinoid reuptake inhibitor (eCBRI)
Miscellaneous
* Cofactor (see Enzyme cofactors)
  • Precursor (see Amino acids)


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