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Template
:
Sympatholytic antihypertensives
From WikiMD's Medical Encyclopedia
Revision as of 15:31, 8 March 2025 by
Prab
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Sympatholytic
(and closely related)
antihypertensives
(
C02
)
Sympatholytics
(antagonize
α-adrenergic
vasoconstriction
)
Central
α
2
-Adrenergic receptor agonists
*
Clonidine
Guanabenz
Guanfacine
Guanoxabenz
Methyldopa
#
Tiamenidine
‡
Adrenergic release inhibitors
*
Bethanidine
Bretylium
Debrisoquine
Guanadrel
Guanazodine
Guancydine
Guanethidine
Guanoclor
Guanoxan
Imidazoline receptor
agonists
*
Moxonidine
Rilmenidine
Tolonidine
Ganglion-blocking
/
nicotinic antagonists
*
Hexamethonium
‡
Mecamylamine
Pentolinium
Trimethaphan
Peripheral
Indirect
Monoamine oxidase inhibitors
*
Pargyline
‡
VMAT inhibitors
*
Bietaserpine
Deserpidine
Methoserpidine
Reserpine
Syrosingopine
Tyrosine hydroxylase inhibitors
*
Metirosine
Direct
α
1
-Adrenergic receptor blockers
*
Doxazosin
Ketanserin
Indoramin
Prazosin
Trimazosin
Urapidil
Non-selective α-adrenergic receptor blockers
*
Phentolamine
Other
antagonists
Serotonin receptor antagonists
*
Ketanserin
Lidanserin
Endothelin receptor antagonists
(for
PH
)
*
dual
(
Aprocitentan
,
Bosentan
,
Macitentan
(
+tadalafil
),
Riociguat
)
selective
(
Ambrisentan
(
+tadalafil
),
Sitaxentan
,
Sotatercept
)
#
WHO-EM
‡
Withdrawn
from market
Clinical trials
:
†
Phase III
§
Never to phase III
Category
:
Drug templates by ATC