3-Phenylpropanoylfentanyl

A synthetic opioid analgesic

3-Phenylpropanoylfentanyl
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3-Phenylpropanoylfentanyl is a synthetic opioid analgesic that is structurally related to fentanyl. It is part of the class of drugs known as fentanyl analogues, which are designed to mimic the effects of fentanyl, a potent opioid used in pain management and anesthesia.

Chemical structure and properties

3-Phenylpropanoylfentanyl is characterized by its chemical structure, which includes a phenylpropanoyl group attached to the fentanyl backbone. The presence of this group differentiates it from other fentanyl analogues and influences its pharmacological properties.

Pharmacology

As with other opioids, 3-Phenylpropanoylfentanyl acts primarily on the mu-opioid receptor in the central nervous system. This interaction results in analgesic effects, as well as potential side effects such as respiratory depression, sedation, and euphoria. The potency and duration of action of 3-Phenylpropanoylfentanyl can vary depending on its specific chemical modifications compared to fentanyl.

Legal status

Due to its potential for abuse and the risk of overdose, 3-Phenylpropanoylfentanyl is often subject to strict regulatory controls. It may be classified as a controlled substance in many jurisdictions, similar to other fentanyl analogues.

Synthesis

The synthesis of 3-Phenylpropanoylfentanyl involves the modification of the fentanyl molecule to include the phenylpropanoyl group. This process requires advanced knowledge of organic chemistry and is typically conducted in a laboratory setting.

Potential risks and side effects

The use of 3-Phenylpropanoylfentanyl carries significant risks, including the potential for opioid overdose. Symptoms of overdose may include extreme drowsiness, slowed breathing, and loss of consciousness. As with other opioids, there is also a risk of developing opioid use disorder with repeated use.

Related pages

• Fentanyl
• Opioid
• Opioid overdose
• Controlled substance

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  Structure of 3-Phenylpropanoylfentanyl