Acetylmethadol
Synthetic opioid analgesic
| Acetylmethadol | |
|---|---|
| |
| INN | |
| Drug class | |
| Routes of administration | |
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| CAS Number | 509-74-0 |
| PubChem | 5284590 |
| DrugBank | DB01450 |
| ChemSpider | 4447600 |
| KEGG | D02763 |
Acetylmethadol is a synthetic opioid analgesic that is chemically related to methadone. It is used primarily in the treatment of opioid dependence. Acetylmethadol is a racemic mixture, meaning it contains equal parts of two enantiomers, which are mirror images of each other.
Pharmacology
Acetylmethadol acts as an agonist at the mu-opioid receptor, which is responsible for its analgesic and euphoric effects. It is metabolized in the liver to form LAAM (levo-alpha-acetylmethadol), which is also an active opioid agonist. The drug has a long half-life, allowing for less frequent dosing compared to other opioids.
Medical use
Acetylmethadol is used in the management of opioid dependence. It is administered orally and is typically used in a controlled clinical setting. The long duration of action makes it suitable for maintenance therapy, reducing the need for frequent dosing and helping to stabilize patients.
Side effects
Common side effects of acetylmethadol include:
Serious side effects can include respiratory depression, which is a risk with all opioid medications.
Legal status
Acetylmethadol is a controlled substance in many countries due to its potential for abuse and dependence. It is classified under various schedules depending on the jurisdiction.
Related pages
Gallery
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Chemical structure of Acetylmethadol
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