Fenethylline: Difference between revisions

From WikiMD's Wellness Encyclopedia

CSV import
Tags: mobile edit mobile web edit
CSV import
 
Line 48: Line 48:
[[Category:Controlled substances]]
[[Category:Controlled substances]]
[[Category:Drugs with no legal status]]
[[Category:Drugs with no legal status]]
<gallery>
File:Fenethylline.svg|Fenethylline
File:Captagon molecule spacefill.png|Fenethylline
</gallery>

Latest revision as of 01:06, 20 February 2025

A synthetic stimulant drug


Fenethylline
INN
Drug class
Routes of administration
Pregnancy category
Bioavailability
Metabolism
Elimination half-life
Excretion
Legal status
CAS Number 3736-08-1
PubChem 8288
DrugBank
ChemSpider 7987
KEGG D07966


Fenethylline, also known as fenetylline and by the brand name Captagon, is a synthetic stimulant that was first synthesized in the 1960s. It is a combination of amphetamine and theophylline, and it was originally used as a treatment for conditions such as attention deficit hyperactivity disorder (ADHD) and narcolepsy.

Pharmacology[edit]

Fenethylline is metabolized by the body into its active components, amphetamine and theophylline. Amphetamine is a potent central nervous system stimulant that increases the release of neurotransmitters such as dopamine and norepinephrine, leading to increased alertness, concentration, and energy. Theophylline is a methylxanthine drug that acts as a bronchodilator and has mild stimulant effects.

Medical Use[edit]

Originally, fenethylline was prescribed for the treatment of ADHD, narcolepsy, and, in some cases, depression. It was favored for its perceived lower side effect profile compared to other stimulants. However, due to its potential for abuse and addiction, fenethylline was eventually banned in most countries.

Abuse and Illicit Use[edit]

Fenethylline has gained notoriety as a drug of abuse, particularly in the Middle East. It is often manufactured illegally and sold under the brand name Captagon. The drug is popular among certain groups due to its ability to enhance physical performance and reduce fatigue, making it a drug of choice in conflict zones.

Legal Status[edit]

Fenethylline is classified as a controlled substance in many countries. It is listed as a Schedule I drug under the United Nations Convention on Psychotropic Substances, indicating that it is considered to have a high potential for abuse and no accepted medical use.

Synthesis[edit]

The synthesis of fenethylline involves the chemical combination of amphetamine and theophylline. The process requires careful control of reaction conditions to ensure the correct formation of the compound. Due to its potential for abuse, the synthesis of fenethylline is heavily regulated.

Related pages[edit]