3-Methylbutyrfentanyl
Synthetic opioid analgesic
| 3-Methylbutyrfentanyl | |
|---|---|
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| CAS Number | 14188-81-9 |
| PubChem | 44469364 |
| DrugBank | |
| ChemSpider | 23274847 |
| KEGG | |
3-Methylbutyrfentanyl is a synthetic opioid analgesic that is an analog of fentanyl. It is a potent agonist of the mu-opioid receptor, similar to other fentanyl analogs, and is used in research settings to study the effects of opioid receptor activation.
Chemical structure and properties
3-Methylbutyrfentanyl is chemically similar to fentanyl, with the primary difference being the substitution of a 3-methylbutyryl group for the propionyl group found in fentanyl. This modification results in changes to its pharmacokinetic and pharmacodynamic properties.
Pharmacology
As a potent mu-opioid receptor agonist, 3-Methylbutyrfentanyl produces effects typical of opioids, including analgesia, euphoria, sedation, and respiratory depression. The potency and efficacy of 3-Methylbutyrfentanyl in activating the mu-opioid receptor are comparable to those of fentanyl, making it a subject of interest in opioid research.
Legal status
Due to its structural similarity to fentanyl and its potential for abuse, 3-Methylbutyrfentanyl is classified as a controlled substance in many jurisdictions. It is often regulated under analog laws that control substances similar to those already scheduled.
Synthesis
The synthesis of 3-Methylbutyrfentanyl involves the acylation of the piperidine nitrogen in the fentanyl structure with 3-methylbutyryl chloride. This chemical reaction is typically carried out under controlled laboratory conditions due to the potency and potential hazards associated with fentanyl analogs.
Related compounds
See also
Gallery
Chemical structure of 3-Methylbutyrfentanyl
3-Methylbutyrfentanyl
Structure of 3-Methylbutyrfentanyl
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Contributors: Prab R. Tumpati, MD
