Trestolone enanthate: Difference between revisions

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Trestolone Enanthate

Trestolone enanthate is a synthetic anabolic-androgenic steroid (AAS) and a derivative of nandrolone. It is an ester of trestolone, also known as 7_-methyl-19-nortestosterone (MENT), and is used in the field of hormone replacement therapy and bodybuilding.

Chemical Structure and Properties

Trestolone enanthate is characterized by the presence of an enanthate ester attached to the 17-beta hydroxyl group of the trestolone molecule. This modification allows for a slower release of the active hormone into the bloodstream, providing a more sustained effect compared to the non-esterified form. The chemical structure of trestolone enanthate can be represented as follows:

Pharmacology

Trestolone enanthate acts as a potent agonist of the androgen receptor, which is responsible for its anabolic and androgenic effects. It is known for its ability to promote muscle growth and increase strength, making it popular among athletes and bodybuilders. Unlike testosterone, trestolone does not undergo 5-alpha reduction to dihydrotestosterone (DHT), which reduces the risk of certain androgenic side effects.

Medical Uses

Trestolone enanthate has been investigated for use in male contraception due to its ability to suppress spermatogenesis while maintaining androgenic activity. It has also been studied for its potential in hormone replacement therapy for men with low testosterone levels.

Side Effects

As with other anabolic steroids, the use of trestolone enanthate can lead to a range of side effects. These may include gynecomastia, acne, hair loss, and liver toxicity. Long-term use can also result in cardiovascular issues and changes in cholesterol levels.

Legal Status

The legal status of trestolone enanthate varies by country. In some regions, it is classified as a controlled substance and is only available by prescription for specific medical conditions. In others, it may be available for research purposes or as a supplement.

Related Pages

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-'''Trestolone enanthate''' is a synthetic and injected anabolic–androgenic steroid (AAS) and a derivative of [[nandrolone]] which was never marketed. It is an androgen ester – specifically, the C17β enanthate ester of [[trestolone]] (7α-methyl-19-nortestosterone; MENT).
+== Trestolone Enanthate ==
-==Pharmacology==
+'''Trestolone enanthate''' is a synthetic anabolic-androgenic steroid (AAS) and a derivative of nandrolone. It is an ester of [[trestolone]], also known as 7_-methyl-19-nortestosterone (MENT), and is used in the field of [[hormone replacement therapy]] and [[bodybuilding]].
-As an [[AAS]], trestolone enanthate is an [[agonist]] of the [[androgen receptor]] (AR), the biological target of androgens like [[testosterone]] and [[dihydrotestosterone]] (DHT). It has strong anabolic effects and weak androgenic effects, which give it a mild side effect profile and make it especially suitable for use in women. The drug has no estrogenic effects but can have progestogenic effects, which can mimic estrogenic side effects.
-==Chemistry==
+== Chemical Structure and Properties ==
-Trestolone enanthate, also known as 7α-methyl-19-nortestosterone 17β-enanthate, is a synthetic [[estrane]] steroid and a derivative of [[nandrolone]]. It is more specifically a derivative of [[19-nortestosterone]] and is a member of the estrane group, while a derivative of [[17β-hydroxyestra-4,9,11-trien-3-one]] (trenbolone), a derivative of [[progesterone]], is a member of the [[estratetraene]] group.
+Trestolone enanthate is characterized by the presence of an enanthate ester attached to the 17-beta hydroxyl group of the trestolone molecule. This modification allows for a slower release of the active hormone into the bloodstream, providing a more sustained effect compared to the non-esterified form. The chemical structure of trestolone enanthate can be represented as follows:
-==History==
+[[File:Trestolone_enanthate.svg|thumb|Chemical structure of Trestolone Enanthate]]
-Trestolone enanthate was first described in the literature in 1963. It was studied for use in male hormonal contraception and treatment of male hypogonadism but was never marketed.
-==Society and culture==
+== Pharmacology ==
-Trestolone enanthate is not currently approved for medical use and it is not available as a prescription medication. However, it has been sold on the internet as a designer steroid for bodybuilders and other athletes.
+Trestolone enanthate acts as a potent agonist of the [[androgen receptor]], which is responsible for its anabolic and androgenic effects. It is known for its ability to promote muscle growth and increase strength, making it popular among athletes and bodybuilders. Unlike testosterone, trestolone does not undergo 5-alpha reduction to dihydrotestosterone (DHT), which reduces the risk of certain androgenic side effects.
-==See also==
+== Medical Uses ==
-* [[List of androgen esters]]
+Trestolone enanthate has been investigated for use in [[male contraception]] due to its ability to suppress [[spermatogenesis]] while maintaining androgenic activity. It has also been studied for its potential in [[hormone replacement therapy]] for men with low testosterone levels.
-* [[List of androgen esters § Trestolone esters]]
-[[Category:Androgens and anabolic steroids]]
+== Side Effects ==
-[[Category:Androgen esters]]
+As with other anabolic steroids, the use of trestolone enanthate can lead to a range of side effects. These may include [[gynecomastia]], [[acne]], [[hair loss]], and [[liver toxicity]]. Long-term use can also result in cardiovascular issues and changes in cholesterol levels.
-[[Category:Estranes]]
-[[Category:Progestogen esters]]
+== Legal Status ==
-{{Anabolic-androgenic steroids}}
+The legal status of trestolone enanthate varies by country. In some regions, it is classified as a controlled substance and is only available by prescription for specific medical conditions. In others, it may be available for research purposes or as a supplement.
-{{Androgen ester stub}}
+== Related Pages ==
+* [[Anabolic steroid]]
+* [[Hormone replacement therapy]]
+* [[Male contraception]]
+[[Category:Anabolic steroids]]