EZH2

From WikiMD.org
Jump to navigation Jump to search

EZH2

EZH2 (pronounced "E-Z-H-two"), also known as Enhancer of Zeste Homolog 2, is a gene that encodes a member of the Polycomb-group (PcG) family. The PcG family has been shown to play a critical role in cancer, epigenetics, and cell differentiation.

Etymology

The name EZH2 stands for "Enhancer of Zeste 2 Polycomb Repressive Complex 2 Subunit". The term "Zeste" is derived from a Drosophila gene, which was found to enhance the expression of the white gene in combination with other mutations. The number "2" indicates that it is the second identified member of this gene family.

Function

EZH2 is part of the Polycomb Repressive Complex 2 (PRC2), which functions in the methylation of Histone H3 on lysine 27 (H3K27), leading to transcriptional repression of the affected target gene. This process is crucial for maintaining cellular differentiation and preventing oncogenesis.

Clinical Significance

Mutations in EZH2 are associated with several types of cancer, including breast, prostate, and non-Hodgkin lymphoma. EZH2 inhibitors are currently being investigated as potential cancer therapeutics.

Related Terms

External links

Esculaap.svg

This WikiMD article is a stub. You can help make it a full article.


Languages: - East Asian 中文, 日本, 한국어, South Asian हिन्दी, Urdu, বাংলা, తెలుగు, தமிழ், ಕನ್ನಡ,
Southeast Asian Indonesian, Vietnamese, Thai, မြန်မာဘာသာ, European español, Deutsch, français, русский, português do Brasil, Italian, polski