Thiorphan

Thiorphan is an enzyme inhibitor that targets enkephalinase, a type of enzyme that breaks down certain peptides in the body. It is primarily used in scientific research to study the effects of these peptides.

Overview

Thiorphan is a potent inhibitor of the enzyme enkephalinase, which is responsible for the degradation of enkephalins in the body. Enkephalins are peptides that play key roles in a variety of physiological processes, including pain perception and mood regulation. By inhibiting enkephalinase, thiorphan increases the levels of enkephalins in the body, which can have a variety of effects.

Uses

Thiorphan is primarily used in scientific research. It is often used in studies investigating the role of enkephalins in the body, as well as the potential therapeutic effects of enkephalinase inhibitors. For example, it has been used in research on pain management, depression, and neurological disorders.

Mechanism of Action

Thiorphan works by binding to the active site of enkephalinase, preventing it from breaking down enkephalins. This increases the levels of enkephalins in the body, which can have a variety of effects depending on the specific enkephalin and its role in the body.

Side Effects

As a research chemical, thiorphan is not typically used in humans, so its side effects are not well-studied. However, because it increases the levels of enkephalins in the body, it could potentially have side effects related to these peptides. For example, it could potentially cause nausea, vomiting, or changes in mood.

See Also

• Enkephalin
• Enzyme inhibitor
• Peptide

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