Solabegron: Difference between revisions

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'''Solabegron''' is a [[beta3-adrenergic receptor]] agonist that is currently under development for the treatment of [[overactive bladder]] and [[irritable bowel syndrome]]. It was initially developed by [[Arena Pharmaceuticals]] and is now being developed by [[Velicept Therapeutic]].
{{DISPLAYTITLE:Solabegron}}


== History ==
== Overview ==
Solabegron was first developed by Arena Pharmaceuticals. In 2013, Arena Pharmaceuticals granted exclusive worldwide rights to develop and commercialize Solabegron to [[Eisai Co.]], Ltd. However, in 2016, Velicept Therapeutic acquired the rights to Solabegron from Eisai Co., Ltd.
'''Solabegron''' is a selective [[beta-3 adrenergic receptor]] agonist that is primarily investigated for its potential therapeutic effects in treating [[overactive bladder]] (OAB) and other related conditions. It is a novel compound that acts by stimulating the beta-3 adrenergic receptors in the bladder, leading to relaxation of the detrusor muscle and increased bladder capacity.


== Mechanism of Action ==
== Mechanism of Action ==
Solabegron works by stimulating the beta3-adrenergic receptors in the bladder, which leads to relaxation of the bladder muscles. This helps to reduce the frequency of urination and the urgency to urinate, which are common symptoms of overactive bladder.
Solabegron works by targeting the [[beta-3 adrenergic receptor]]s located in the bladder. Activation of these receptors results in the relaxation of the detrusor muscle, which is the smooth muscle found in the wall of the bladder. This relaxation helps to increase the bladder's capacity to hold urine and reduces the symptoms of urgency and frequency associated with [[overactive bladder]].


== Clinical Trials ==
== Clinical Applications ==
Several clinical trials have been conducted to evaluate the safety and efficacy of Solabegron. In a Phase 2 trial, Solabegron was found to be effective in reducing the symptoms of overactive bladder. A Phase 3 trial is currently underway.
The primary clinical application of solabegron is in the management of [[overactive bladder]], a condition characterized by a sudden, involuntary contraction of the muscle in the wall of the urinary bladder, leading to an urgent need to urinate. Solabegron is being studied for its potential to provide relief from the symptoms of OAB without the side effects commonly associated with other treatments, such as [[anticholinergic]] medications.


== Potential Side Effects ==
== Development and Research ==
As with any medication, Solabegron may cause side effects. The most common side effects reported in clinical trials include headache, urinary tract infection, and dry mouth. However, these side effects were generally mild and did not lead to discontinuation of the medication.
Solabegron is currently under investigation in various clinical trials to assess its efficacy and safety profile. Early studies have shown promising results, indicating that solabegron may be effective in reducing the symptoms of [[overactive bladder]] with a favorable side effect profile. Ongoing research aims to further establish its role in the treatment of OAB and potentially other conditions involving smooth muscle relaxation.


== See Also ==
== Side Effects ==
* [[Beta3-adrenergic receptor]]
As with any medication, solabegron may have side effects. Commonly reported side effects include headache, nausea, and dizziness. However, it is generally well-tolerated, and the incidence of side effects is lower compared to traditional [[anticholinergic]] therapies used for [[overactive bladder]].
 
== Future Directions ==
Research is ongoing to explore additional therapeutic uses of solabegron beyond [[overactive bladder]]. Potential areas of interest include its application in treating [[irritable bowel syndrome]] and other conditions where smooth muscle relaxation may be beneficial. Further studies are needed to fully understand the scope of solabegron's therapeutic potential.
 
== Related Pages ==
* [[Overactive bladder]]
* [[Overactive bladder]]
* [[Beta-3 adrenergic receptor]]
* [[Anticholinergic]]
* [[Irritable bowel syndrome]]
* [[Irritable bowel syndrome]]
* [[Arena Pharmaceuticals]]
* [[Velicept Therapeutic]]


[[Category:Drugs]]
[[File:Solabegron.svg|thumb|right|Chemical structure of Solabegron]]
[[Category:Pharmaceuticals]]
[[Category:Medicine]]


{{stub}}
[[Category:Beta-3 adrenergic receptor agonists]]
[[Category:Experimental drugs]]

Latest revision as of 03:45, 13 February 2025


Overview[edit]

Solabegron is a selective beta-3 adrenergic receptor agonist that is primarily investigated for its potential therapeutic effects in treating overactive bladder (OAB) and other related conditions. It is a novel compound that acts by stimulating the beta-3 adrenergic receptors in the bladder, leading to relaxation of the detrusor muscle and increased bladder capacity.

Mechanism of Action[edit]

Solabegron works by targeting the beta-3 adrenergic receptors located in the bladder. Activation of these receptors results in the relaxation of the detrusor muscle, which is the smooth muscle found in the wall of the bladder. This relaxation helps to increase the bladder's capacity to hold urine and reduces the symptoms of urgency and frequency associated with overactive bladder.

Clinical Applications[edit]

The primary clinical application of solabegron is in the management of overactive bladder, a condition characterized by a sudden, involuntary contraction of the muscle in the wall of the urinary bladder, leading to an urgent need to urinate. Solabegron is being studied for its potential to provide relief from the symptoms of OAB without the side effects commonly associated with other treatments, such as anticholinergic medications.

Development and Research[edit]

Solabegron is currently under investigation in various clinical trials to assess its efficacy and safety profile. Early studies have shown promising results, indicating that solabegron may be effective in reducing the symptoms of overactive bladder with a favorable side effect profile. Ongoing research aims to further establish its role in the treatment of OAB and potentially other conditions involving smooth muscle relaxation.

Side Effects[edit]

As with any medication, solabegron may have side effects. Commonly reported side effects include headache, nausea, and dizziness. However, it is generally well-tolerated, and the incidence of side effects is lower compared to traditional anticholinergic therapies used for overactive bladder.

Future Directions[edit]

Research is ongoing to explore additional therapeutic uses of solabegron beyond overactive bladder. Potential areas of interest include its application in treating irritable bowel syndrome and other conditions where smooth muscle relaxation may be beneficial. Further studies are needed to fully understand the scope of solabegron's therapeutic potential.

Related Pages[edit]

Chemical structure of Solabegron